From: Dual EZH2 and EHMT2 histone methyltransferase inhibition increases biological efficacy in breast cancer cells
Cell growth assay (IC50 μM)
HKMT-1-005
BIX-01294
UNC0638
GSK343
Cell viability (MTT)
4.3
9.6
8.2
>15
Clonogenic
0.41
1.4
1.1
>50